As a leading (3S)-10-(1-Aminocyclopropyl)-9-Fluoro-2,3-Dihydro-3-Methyl-7-Oxo-7H-Pyrido[1,2,3-De]-1,4-Benzoxazine-6-Carboxylic Acid Methanesulfonate supplier, we deliver high-quality products across diverse grades to meet evolving needs, empowering global customers with safe, efficient, and compliant chemical solutions.
What is the chemical structure of (3S) -10- (1-aminocyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylic acid methanesulfonate
The chemical structure of (3S) -10- (1-hydroxycyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-ethyl carboxylate is like a delicate mechanism, which is cleverly linked by various atoms in a specific order and spatial relationship.
This structure is based on [1,2,3-De] -1,4-benzoxazine as the core parent ring, which is like the foundation of a pavilion and lays the molecular structure. Above the parent ring, there are ethyl carboxylate groups at the 6-position, such as building cornices, which endow the molecule with specific reactivity and properties. The 7-position oxygen atom forms a carbonyl group, which is a key activity check point and has a profound impact on molecular reactivity.
3-position methyl groups are like wind chimes under the eaves. Although they are small, they have subtle effects on molecular spatial steric resistance and physicochemical properties. 2,3-dihydrogen indicates that this segment of the structure contains partially saturated carbon-carbon bonds, which affects molecular flexibility and stability. The 9-position fluorine atom resembles a hidden mechanism, which significantly changes the distribution of molecular electron clouds, affecting lipophilicity and biological activity.
10-position continuous (1-hydroxy cyclopropyl), such as delicate accessories, hydroxyl groups are active and reactive, and the special tension of cyclopropyl groups affects the overall activity and configuration of molecules. Such various structural fragments cooperate with each other to form a unique and complex chemical structure, which is the source of the unique physicochemical and biological activities of the compound.
What is the main use of (3S) -10- (1-aminocyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylic acid methanesulfonate?
What are the main uses of (3S) -10- (1-hydroxycyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylic acid methyl ester?
(3S) -10- (1-hydroxycyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylic acid methyl ester, such compounds have important uses in the field of medicine. Its structural properties give it unique pharmacological activity.
It has shown significant efficacy in the development of antibacterial drugs. With its special molecular configuration, it can effectively inhibit the growth and reproduction of a variety of bacteria. It has inhibitory effects on common Gram-positive and Gram-negative bacteria, such as Escherichia coli, Staphylococcus aureus, etc. Its mechanism of action is to interfere with the normal metabolic process of bacteria through a specific chemical structure combined with key targets inside the bacteria, so as to achieve the purpose of antibacterial.
In addition, the compound has also emerged in the treatment of some infectious diseases. Due to its ability to precisely act on pathogens that cause infections, it is expected to become a key component of new anti-infective drugs, providing new and effective means for the clinical treatment of infectious diseases, helping to solve the current problem of antimicrobial resistance, and bringing new treatment hope to patients.
What is the pharmacological mechanism of (3S) -10- (1-aminocyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylate methanesulfonate?
The pharmacological mechanism of (3S) -10- (1-hydroxycyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylate methyl ester is really an interesting topic. The mechanism of action of this drug is like a delicate mechanism, which is interconnected and exerts unique effects in the microscopic environment.
From a molecular perspective, specific groups in its structure, such as the (3S) configuration part, give the molecule a specific spatial orientation, which is like a precise key to fit the keyhole of a specific biological target. 1-Hydroxycyclopropyl may stabilize the drug-target complex and enhance the binding affinity by interacting with specific regions of the target, such as hydrogen bonds.
The introduction of 9-fluorine atoms significantly changes the electron cloud distribution of the molecule, which in turn affects its lipid solubility and chemical reactivity. This property may help the drug to cross the biofilm and reach the target efficiently, or change the binding force to the target, optimizing pharmacological activity.
Furthermore, the complex parent nuclear structure of 2,3-dihydro-3-methyl-7-oxo-7H-pyrido [1,2,3-De] -1,4-benzoxazine-6-methyl carboxylate is like a fully functional castle. The structure of pyridyl-benzoxazine provides a rigid plane, which is conducive to the formation of π-π stacking and other interactions with the target, while the methyl carboxylate group, or participates in the ion-dipole, hydrogen bond and other forces of the target, together to build a stable binding mode.
In summary, this drug precisely acts on specific biological targets through a variety of intermolecular forces through its unique chemical structure and regulates related biological processes to achieve specific pharmacological effects. It is a masterpiece carefully crafted in the field of pharmacy.
What are the side effects of (3S) -10- (1-aminocyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylate methanesulfonate
(3S) -10- (1-hydroxycyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylate methyl ester, the side effects of this substance are various.
It may cause gastrointestinal discomfort, such as nausea, vomiting, abdominal pain, diarrhea, etc. This reaction is caused by the drug entering the body, irritating the gastrointestinal mucosa and disturbing the normal transportation and transformation of the gastrointestinal tract.
It may also affect the central nervous system, such as headache, dizziness, insomnia, and even cause mental abnormalities. This condition occurs because drugs can penetrate the blood-brain barrier and interfere with the transmission of neurotransmitters and the normal function of the nervous system.
And it also has potential effects on the liver, kidneys and other organs. The liver is the official for detoxification, and the kidneys are responsible for excretion. The metabolism of drugs through these two organs may increase their burden, affect their normal function, and cause abnormal liver and kidney function indicators.
It may also cause allergic reactions, such as rash, itching, severe cases, or anaphylactic shock. This is caused by an excessive immune response to drug ingredients by the individual's immune system. When using medication, when carefully observing to pay attention to whether there are such side effects. If there is any abnormality, it is advisable to seek medical treatment immediately to ensure the safety of medication.
What is the market prospect of (3S) -10- (1-aminocyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylic acid methanesulfonate?
What is the market prospect of (3S) -10- (1-hydroxycyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyridino [1,2,3-De] -1,4-benzoxazine-6-carboxylic acid methyl ester? I will take the ancient saying of "Tiangong Kaiwu" as your solution.
Looking at this compound, its unique structure and fusion of various groups seem to contain the wonders of creation. Hydroxycyclopropyl, fluorine atoms, methyl groups, etc. are in their respective positions and interact, giving them unique chemical properties and potential activities.
In the field of medicine, these structures may bring opportunities for the creation of new drugs. Nowadays, there are many kinds of diseases, and the demand for medicine is eager. If it can demonstrate good pharmacological activity and exert curative effect on specific diseases, it will surely rise like a surprise and win a place in the market.
Looking at the road of scientific research and exploration, chemists have never stopped studying new compounds. If this compound shows good drug potential in the laboratory and is verified by clinical trials, once it is approved to enter the market, the prospects are limitless.
However, the road to the market is not smooth. New drug research and development is expensive and time-consuming, like a long journey, requiring a lot of manpower, material resources and financial investment. And competition is fierce, many pharmaceutical companies are coveting the fertile soil of the pharmaceutical market, and there are many new ones. If you want to stand out, you need to have excellent efficacy, safety and reasonable price.
Furthermore, the impact of policies and regulations cannot be ignored. Drug approval is strict, and only those in compliance can enter the market. Therefore, if we can make good use of our unique structural advantages, conform to the trend of pharmaceutical development, and meet the challenges of all parties, this (3S) -10- (1-hydroxycyclopropyl) -9-fluoro-2,3-dihydro-3-methyl-7-oxo-7H-pyrido [1,2,3-De] -1,4-benzoxazine-6-carboxylate methyl ester may bloom in the market, adding to the pharmaceutical industry and benefiting patients.